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دواعي استعمال اكنيتون 5مجم/مل 5 امبول

معلومات من نشرات دوائية ومراجع موثقة، مع مصدر كل معلومة. السعر الحالي: 60ج.م.

عن الدواء

Akineton 5 mg/ml injection, 5 ampoules (biperiden lactate).

دواعي الاستعمال
  • All forms of parkinsonism (injection especially when rapid onset is needed or for initial therapy in severe cases).الفئة: AdultsBASG (Austrian Federal Office for Safety in Health Care) medicines database
  • Drug-induced extrapyramidal symptoms (e.g. acute dystonia, akathisia, parkinsonoid, rigidity).الفئة: Adults and childrenBASG (Austrian Federal Office for Safety in Health Care) medicines database
  • Nicotine poisoning and organophosphate poisoning.الفئة: AdultsBASG (Austrian Federal Office for Safety in Health Care) medicines database
الآثار الجانبية
  • Rare: restlessness, agitation, confusion, hallucinations at higher doses, fatigue, dizziness, memory disturbance, tachycardia, dry mouth, nausea, muscle twitching. Very rare: hypersensitivity, accommodation disorders, mydriasis, bradycardia, constipation, micturition disorders; hypotension possible after parenteral use.نشرة دولية لنفس المنتج · BASG (Austrian Federal Office for Safety in Health Care) medicines database
موانع الاستعمال
  • Hypersensitivity to biperiden or excipients; untreated narrow-angle glaucoma; mechanical stenosis of the GI tract; megacolon; ileus.نشرة دولية لنفس المنتج · BASG (Austrian Federal Office for Safety in Health Care) medicines database
تحذيرات واحتياطات
  • May lower seizure threshold; caution in prostatic hypertrophy (urinary retention), glaucoma (monitor intraocular pressure), myasthenia gravis and conditions causing tachycardia; elderly with organic brain disease more sensitive; memory impairment, abuse potential; avoid abrupt withdrawal; may impair driving.نشرة دولية لنفس المنتج · BASG (Austrian Federal Office for Safety in Health Care) medicines database
التداخلات الدوائية
  • Other anticholinergic drugs (psychotropics, antihistamines, antiparkinson agents, spasmolytics)Increased central and peripheral anticholinergic effects.BASG (Austrian Federal Office for Safety in Health Care) medicines database
  • QuinidineEnhanced anticholinergic cardiovascular effects (AV conduction).BASG (Austrian Federal Office for Safety in Health Care) medicines database
  • LevodopaDyskinesias may be increased.BASG (Austrian Federal Office for Safety in Health Care) medicines database
  • AlcoholAlcohol effect may be increased; avoid alcohol.BASG (Austrian Federal Office for Safety in Health Care) medicines database
  • MetoclopramideGI effects of metoclopramide antagonised.BASG (Austrian Federal Office for Safety in Health Care) medicines database
  • PethidineCNS adverse effects may be increased.BASG (Austrian Federal Office for Safety in Health Care) medicines database
الحمل والرضاعة
  • Use in pregnancy only after careful benefit-risk assessment; no experience in pregnancy.نشرة دولية لنفس المنتج · BASG (Austrian Federal Office for Safety in Health Care) medicines database
  • Anticholinergics may inhibit lactation and biperiden probably passes into milk; breastfeeding should be stopped.نشرة دولية لنفس المنتج · BASG (Austrian Federal Office for Safety in Health Care) medicines database
المتابعة أثناء العلاج
  • Check intraocular pressure regularly.نشرة دولية لنفس المنتج · BASG (Austrian Federal Office for Safety in Health Care) medicines database
كيف يعمل الدواء
  • بيبيريدين لاكتات: Predominantly central anticholinergic; binds competitively to central and peripheral muscarinic (mainly M1) receptors.مضاد للكولين مركزي التأثير (مضاد لمستقبلات المسكارين)

المصادر