دواعي استعمال اكنيتون 5مجم/مل 5 امبول
معلومات من نشرات دوائية ومراجع موثقة، مع مصدر كل معلومة. السعر الحالي: 60ج.م.
عن الدواء
Akineton 5 mg/ml injection, 5 ampoules (biperiden lactate).
دواعي الاستعمال
- All forms of parkinsonism (injection especially when rapid onset is needed or for initial therapy in severe cases).الفئة: AdultsBASG (Austrian Federal Office for Safety in Health Care) medicines database
- Drug-induced extrapyramidal symptoms (e.g. acute dystonia, akathisia, parkinsonoid, rigidity).الفئة: Adults and childrenBASG (Austrian Federal Office for Safety in Health Care) medicines database
- Nicotine poisoning and organophosphate poisoning.الفئة: AdultsBASG (Austrian Federal Office for Safety in Health Care) medicines database
الآثار الجانبية
- Rare: restlessness, agitation, confusion, hallucinations at higher doses, fatigue, dizziness, memory disturbance, tachycardia, dry mouth, nausea, muscle twitching. Very rare: hypersensitivity, accommodation disorders, mydriasis, bradycardia, constipation, micturition disorders; hypotension possible after parenteral use.نشرة دولية لنفس المنتج · BASG (Austrian Federal Office for Safety in Health Care) medicines database
موانع الاستعمال
- Hypersensitivity to biperiden or excipients; untreated narrow-angle glaucoma; mechanical stenosis of the GI tract; megacolon; ileus.نشرة دولية لنفس المنتج · BASG (Austrian Federal Office for Safety in Health Care) medicines database
تحذيرات واحتياطات
- May lower seizure threshold; caution in prostatic hypertrophy (urinary retention), glaucoma (monitor intraocular pressure), myasthenia gravis and conditions causing tachycardia; elderly with organic brain disease more sensitive; memory impairment, abuse potential; avoid abrupt withdrawal; may impair driving.نشرة دولية لنفس المنتج · BASG (Austrian Federal Office for Safety in Health Care) medicines database
التداخلات الدوائية
- Other anticholinergic drugs (psychotropics, antihistamines, antiparkinson agents, spasmolytics)Increased central and peripheral anticholinergic effects.BASG (Austrian Federal Office for Safety in Health Care) medicines database
- QuinidineEnhanced anticholinergic cardiovascular effects (AV conduction).BASG (Austrian Federal Office for Safety in Health Care) medicines database
- LevodopaDyskinesias may be increased.BASG (Austrian Federal Office for Safety in Health Care) medicines database
- AlcoholAlcohol effect may be increased; avoid alcohol.BASG (Austrian Federal Office for Safety in Health Care) medicines database
- MetoclopramideGI effects of metoclopramide antagonised.BASG (Austrian Federal Office for Safety in Health Care) medicines database
- PethidineCNS adverse effects may be increased.BASG (Austrian Federal Office for Safety in Health Care) medicines database
الحمل والرضاعة
- Use in pregnancy only after careful benefit-risk assessment; no experience in pregnancy.نشرة دولية لنفس المنتج · BASG (Austrian Federal Office for Safety in Health Care) medicines database
- Anticholinergics may inhibit lactation and biperiden probably passes into milk; breastfeeding should be stopped.نشرة دولية لنفس المنتج · BASG (Austrian Federal Office for Safety in Health Care) medicines database
المتابعة أثناء العلاج
- Check intraocular pressure regularly.نشرة دولية لنفس المنتج · BASG (Austrian Federal Office for Safety in Health Care) medicines database
كيف يعمل الدواء
- بيبيريدين لاكتات: Predominantly central anticholinergic; binds competitively to central and peripheral muscarinic (mainly M1) receptors.مضاد للكولين مركزي التأثير (مضاد لمستقبلات المسكارين)
المصادر
- السعر: قوائم أسعار الأدوية المنشورة في مصر.
- BASG (Austrian Federal Office for Safety in Health Care) medicines database