دواعي استعمال تاكيبريل 100 مجم/5مل حقن في القراب
معلومات من نشرات دوائية ومراجع موثقة، مع مصدر كل معلومة. السعر الحالي: 45ج.م.
عن الدواء
Hyperbaric prilocaine hydrochloride 100 mg/5 ml (2%) solution for intrathecal (spinal) injection, 1 ampoule; Sintetica GmbH, marketed via Sunny Medical/Sunny Pharma.
دواعي الاستعمال
- Spinal anaesthesia in adults for short-term surgical proceduresالفئة: Adultselectronic medicines compendium (emc), UK
الآثار الجانبية
- Effects similar to other spinal amide anaesthetics: hypotension, bradycardia, paraesthesia, dizziness, nausea; rarely methaemoglobinaemia/cyanosis, allergic reactions, CNS toxicity signs; post-spinal headache.نشرة دولية لنفس التركيبة · electronic medicines compendium (emc), UK
موانع الاستعمال
- Hypersensitivity to prilocaine or other amide local anaesthetics; serious cardiac conduction problems; severe anaemia; decompensated cardiac insufficiency; cardiogenic or hypovolaemic shock; congenital or acquired methaemoglobinaemia; concomitant anticoagulant therapy; general contraindications to subarachnoid anaesthesia; children under 6 months; injection into infected areas.نشرة دولية لنفس التركيبة · electronic medicines compendium (emc), UK
تحذيرات واحتياطات
- Risk of methaemoglobinaemia (potentiated by methaemoglobin-inducing drugs); caution in heart block, cardiac decompensation, advanced liver or kidney damage and the elderly.نشرة دولية لنفس التركيبة · electronic medicines compendium (emc), UK
التداخلات الدوائية
- Methaemoglobin-inducing drugs (sulfonamides, antimalarials, sodium nitroprusside, nitroglycerin)May potentiate methaemoglobin formation.electronic medicines compendium (emc), UK
- Other local anaesthetics and structurally similar antiarrhythmics (lidocaine, mexiletine, tocainide); class III antiarrhythmicsAdditive undesirable effects; caution.electronic medicines compendium (emc), UK
الحمل والرضاعة
- No adequate human data; prilocaine crosses the placenta; neonatal methaemoglobinaemia reported after paracervical/pudendal obstetric use; use only with a compelling indication.نشرة دولية لنفس التركيبة · electronic medicines compendium (emc), UK
- Unknown whether excreted in milk; breastfeeding can be resumed about 24 hours after treatment.نشرة دولية لنفس التركيبة · electronic medicines compendium (emc), UK
كيف يعمل الدواء
- بريلوكائين: مخدر موضعي من الأميدات
المصادر
- السعر: قوائم أسعار الأدوية المنشورة في مصر.
- electronic medicines compendium (emc), UK
- WHO Collaborating Centre for Drug Statistics Methodology